Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles

The reactions of 4-R- and 6-R-2-nitroanisoles (R = Me, Br) in neat cyclohexylamine and piperidine have been studied. The reactions with cyclohexylamine lead to the respective aromatic nucleophilic substitution products while the reactions with piperidine mainly yield the substituted nitrophenols. It...

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Autores principales: Nudelman, N.S., Palleros, D.R.
Formato: JOUR
Acceso en línea:http://hdl.handle.net/20.500.12110/paper_1472779X_v_n6_p805_Nudelman
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spelling todo:paper_1472779X_v_n6_p805_Nudelman2023-10-03T16:18:03Z Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles Nudelman, N.S. Palleros, D.R. The reactions of 4-R- and 6-R-2-nitroanisoles (R = Me, Br) in neat cyclohexylamine and piperidine have been studied. The reactions with cyclohexylamine lead to the respective aromatic nucleophilic substitution products while the reactions with piperidine mainly yield the substituted nitrophenols. It was found that 6-R-2-nitroanisoles react faster than the respective 4-R-2-nitroanisoles. The absence of the expected primary steric effect is thought to be due to the spatial arrangement of the methoxide group, which adopts a conformation perpendicular to the ring plane when it is surrounded by two ortho-substituents. CNDO and INDO calculations for different conformations of the substrates give support to this assumption. JOUR info:eu-repo/semantics/openAccess http://creativecommons.org/licenses/by/2.5/ar http://hdl.handle.net/20.500.12110/paper_1472779X_v_n6_p805_Nudelman
institution Universidad de Buenos Aires
institution_str I-28
repository_str R-134
collection Biblioteca Digital - Facultad de Ciencias Exactas y Naturales (UBA)
description The reactions of 4-R- and 6-R-2-nitroanisoles (R = Me, Br) in neat cyclohexylamine and piperidine have been studied. The reactions with cyclohexylamine lead to the respective aromatic nucleophilic substitution products while the reactions with piperidine mainly yield the substituted nitrophenols. It was found that 6-R-2-nitroanisoles react faster than the respective 4-R-2-nitroanisoles. The absence of the expected primary steric effect is thought to be due to the spatial arrangement of the methoxide group, which adopts a conformation perpendicular to the ring plane when it is surrounded by two ortho-substituents. CNDO and INDO calculations for different conformations of the substrates give support to this assumption.
format JOUR
author Nudelman, N.S.
Palleros, D.R.
spellingShingle Nudelman, N.S.
Palleros, D.R.
Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
author_facet Nudelman, N.S.
Palleros, D.R.
author_sort Nudelman, N.S.
title Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
title_short Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
title_full Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
title_fullStr Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
title_full_unstemmed Theoretical calculations of chemical interactions. Part 4. Aromatic nucleophilic substitutions and SN2 reactions of 4- and 6-substituted 2-nitroanisoles
title_sort theoretical calculations of chemical interactions. part 4. aromatic nucleophilic substitutions and sn2 reactions of 4- and 6-substituted 2-nitroanisoles
url http://hdl.handle.net/20.500.12110/paper_1472779X_v_n6_p805_Nudelman
work_keys_str_mv AT nudelmanns theoreticalcalculationsofchemicalinteractionspart4aromaticnucleophilicsubstitutionsandsn2reactionsof4and6substituted2nitroanisoles
AT pallerosdr theoreticalcalculationsofchemicalinteractionspart4aromaticnucleophilicsubstitutionsandsn2reactionsof4and6substituted2nitroanisoles
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