Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives

A novel series of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted (3a-p) has been synthesized. The intermediates 2-hydrazolyl-3-phenyl-4-thiazolidinone substituted (2a-p) were prepared by condensation of benzaldehyde 4-phenyl-3-thiosemicarbazone substituted (1a-p) with ethy...

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Autores principales: Góes, Alexandre J. S., Melo, Edésio J.T., Alves, Antonio J., Lima, José G., Araújo, Janete M., Faria, Antônio R., Alves, Anselmo Q., Lima, Vânia T., Carvalho, Cristiane S., Spacov, Isabel C.G., Nascimento, André A.P.L., Aquino, Thiago M.
Formato: Articulo
Lenguaje:Inglés
Publicado: 2011
Materias:
Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/8340
http://www.latamjpharm.org/resumenes/30/8/LAJOP_30_8_1_18.pdf
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id I19-R120-10915-8340
record_format dspace
institution Universidad Nacional de La Plata
institution_str I-19
repository_str R-120
collection SEDICI (UNLP)
language Inglés
topic Farmacia
antimicrobial activity; anti-toxoplasma gondii activity; 4-thiazolidinone; thiosemicarbazone
spellingShingle Farmacia
antimicrobial activity; anti-toxoplasma gondii activity; 4-thiazolidinone; thiosemicarbazone
Góes, Alexandre J. S.
Melo, Edésio J.T.
Alves, Antonio J.
Lima, José G.
Araújo, Janete M.
Faria, Antônio R.
Alves, Anselmo Q.
Lima, Vânia T.
Carvalho, Cristiane S.
Spacov, Isabel C.G.
Nascimento, André A.P.L.
Aquino, Thiago M.
Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
topic_facet Farmacia
antimicrobial activity; anti-toxoplasma gondii activity; 4-thiazolidinone; thiosemicarbazone
description A novel series of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted (3a-p) has been synthesized. The intermediates 2-hydrazolyl-3-phenyl-4-thiazolidinone substituted (2a-p) were prepared by condensation of benzaldehyde 4-phenyl-3-thiosemicarbazone substituted (1a-p) with ethyl chloroacetate. Theses intermediates were submitted to reaction with ethyl 2-cyano-3-(4-nitrophenyl)-acetate to give the title compounds. The 4-thiazolidinones were screened for their anti-Toxoplasma gondii, and all derivatives promoted decrease of percentage of infection of Vero cells, with elimination of intracellular tachyzoites. The LD50 ranged around 0.5 mM for the intracellular parasites and were higher than 10 mM for Vero cells. According to results of antimicrobial activity, only two compounds showed significant inhibition against M. luteus, but demonstrated higher values of MIC and MBC when compared with standard drug.
format Articulo
Articulo
author Góes, Alexandre J. S.
Melo, Edésio J.T.
Alves, Antonio J.
Lima, José G.
Araújo, Janete M.
Faria, Antônio R.
Alves, Anselmo Q.
Lima, Vânia T.
Carvalho, Cristiane S.
Spacov, Isabel C.G.
Nascimento, André A.P.L.
Aquino, Thiago M.
author_facet Góes, Alexandre J. S.
Melo, Edésio J.T.
Alves, Antonio J.
Lima, José G.
Araújo, Janete M.
Faria, Antônio R.
Alves, Anselmo Q.
Lima, Vânia T.
Carvalho, Cristiane S.
Spacov, Isabel C.G.
Nascimento, André A.P.L.
Aquino, Thiago M.
author_sort Góes, Alexandre J. S.
title Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
title_short Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
title_full Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
title_fullStr Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
title_full_unstemmed Synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
title_sort synthesis, anti-toxoplasma gondii and antimicrobial activities of 2-hydrazolyl-3-phenyl-5-(4-nitrobenzylidene)-4-thiazolidinone substituted derivatives
publishDate 2011
url http://sedici.unlp.edu.ar/handle/10915/8340
http://www.latamjpharm.org/resumenes/30/8/LAJOP_30_8_1_18.pdf
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