Preparation, crystal structure and prodrug studies of genistein benzensulfonate
4'-ethyl-7-phenylsulfonylgenistein (EPG, 3), a potential prodrug for genistein (1), was synthesized in high yield and its crystal structure was reported firstly. It possesses better physical and chemical properties such as solubility, lipid/water partition coefficient, LogP, and hydrolysis kine...
Guardado en:
| Autores principales: | Peng, You, Gan, Li- Jun, Deng, Ze-yuan |
|---|---|
| Formato: | Articulo Comunicacion |
| Lenguaje: | Inglés |
| Publicado: |
2011
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| Materias: | |
| Acceso en línea: | http://sedici.unlp.edu.ar/handle/10915/8322 http://www.latamjpharm.org/resumenes/30/7/LAJOP_30_7_2_7.pdf |
| Aporte de: |
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