A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats

A simple HPLC method was developed to study the pharmacokinetics of tobramycin in rat after intravenous administration. The plasma samples were deproteinized with acetonitrile after addition of the internal standard, netilmicin. The separation was achieved on a reversed-phase C18 column after deriva...

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Autores principales: Zhang, Zhenyuan, Peng, Jingdong
Formato: Articulo Comunicacion
Lenguaje:Inglés
Publicado: 2011
Materias:
Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/8180
http://www.latamjpharm.org/resumenes/30/3/LAJOP_30_3_2_5.pdf
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id I19-R120-10915-8180
record_format dspace
institution Universidad Nacional de La Plata
institution_str I-19
repository_str R-120
collection SEDICI (UNLP)
language Inglés
topic Farmacia
Técnicas de Química Analítica
antibiótico
9-fluorenylmerthyl chloroformate; high-performance liquid chromatography; pharmacokinetic study; tobramycin
spellingShingle Farmacia
Técnicas de Química Analítica
antibiótico
9-fluorenylmerthyl chloroformate; high-performance liquid chromatography; pharmacokinetic study; tobramycin
Zhang, Zhenyuan
Peng, Jingdong
A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
topic_facet Farmacia
Técnicas de Química Analítica
antibiótico
9-fluorenylmerthyl chloroformate; high-performance liquid chromatography; pharmacokinetic study; tobramycin
description A simple HPLC method was developed to study the pharmacokinetics of tobramycin in rat after intravenous administration. The plasma samples were deproteinized with acetonitrile after addition of the internal standard, netilmicin. The separation was achieved on a reversed-phase C18 column after derivatization with 9-fluorenylmethyl chloroformate (FMOC-Cl) in borate buffer (0.2 M, pH 6.5) for 15 min at 25 ºC. The mobile phase was water-acetonitrile (6:94, v/v) at a flow rate of 1.0 mL/min. The fluorescence excitation and emission wavelengths were 265 and 315 nm, respectively. The method was linear over the range of 0.12-10.48 μg/mL for tobramycin in plasma. The limit of detection was 0.074 μg/mL. The intra-day and inter-day precisions of tobramycin were both less than 6%. Both derivatives were stable in the reaction solution for 24 h at room temperature. This assay had been successfully applied to the in vivo kinetic study of tobramycin in rats.
format Articulo
Comunicacion
author Zhang, Zhenyuan
Peng, Jingdong
author_facet Zhang, Zhenyuan
Peng, Jingdong
author_sort Zhang, Zhenyuan
title A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
title_short A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
title_full A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
title_fullStr A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
title_full_unstemmed A simple HPLC method for determination tobramycin in plasma and Iis application in the study of pharmacokinetics in rats
title_sort simple hplc method for determination tobramycin in plasma and iis application in the study of pharmacokinetics in rats
publishDate 2011
url http://sedici.unlp.edu.ar/handle/10915/8180
http://www.latamjpharm.org/resumenes/30/3/LAJOP_30_3_2_5.pdf
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AT zhangzhenyuan simplehplcmethodfordeterminationtobramycininplasmaandiisapplicationinthestudyofpharmacokineticsinrats
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