Pharmacokinetics, tissue distribution and excretion of Vitexin in mice

Pharmacokinetics, tissue distribution and excretion of vitexin (VIT) were studied after intravenous and oral administration to mice at dose of 10 mg/kg and 30 mg/kg, respectively. A sensitive and specific HPLC method with internal standard was developed and validated for the pharmacokinetic studies...

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Autores principales: Wang, Yun-jiao, Qu, Gong-lin, Zhang, Wen-jie, Xue, He-fei, Chen, Ying-hui, Yin, Jing-jing, Lu, Dong-rui, Ying, Xi-xiang
Formato: Articulo
Lenguaje:Inglés
Publicado: 2012
Materias:
Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/25695
http://www.latamjpharm.org/resumenes/31/6/LAJOP_31_6_1_8.pdf
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id I19-R120-10915-25695
record_format dspace
institution Universidad Nacional de La Plata
institution_str I-19
repository_str R-120
collection SEDICI (UNLP)
language Inglés
topic Farmacia
Farmacocinética
Distribución Tisular
Cromatografía Líquida de Alta Presión
excretion
Vitexin
spellingShingle Farmacia
Farmacocinética
Distribución Tisular
Cromatografía Líquida de Alta Presión
excretion
Vitexin
Wang, Yun-jiao
Qu, Gong-lin
Zhang, Wen-jie
Xue, He-fei
Chen, Ying-hui
Yin, Jing-jing
Lu, Dong-rui
Ying, Xi-xiang
Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
topic_facet Farmacia
Farmacocinética
Distribución Tisular
Cromatografía Líquida de Alta Presión
excretion
Vitexin
description Pharmacokinetics, tissue distribution and excretion of vitexin (VIT) were studied after intravenous and oral administration to mice at dose of 10 mg/kg and 30 mg/kg, respectively. A sensitive and specific HPLC method with internal standard was developed and validated for the pharmacokinetic studies of VIT. The results showed that VIT was rapidly and widespreadly distributed throughout the whole body after administration and the oral bioavailability of VIT was 3.91 %. The highest VIT level after intravenous dose was obtained in gallbladder, followed by lung, liver and kidney. While, the highest VIT level after oral dose was observed in gallbladder, followed by intestine, stomach, and spleen. The total cumulative excretion percentage of VIT in 24 h after intravenous and oral administration are 31.83 ± 3.85 % (22.72 ± 2.23 % in urinary excretion; 9.11 ± 1.69 % in fecal excretion) and 10.77 ± 2.34 % (2.92 ±1.05 % in urinary excretion; 7.85 ± 1.45 % in fecal excretion), respectively.
format Articulo
Articulo
author Wang, Yun-jiao
Qu, Gong-lin
Zhang, Wen-jie
Xue, He-fei
Chen, Ying-hui
Yin, Jing-jing
Lu, Dong-rui
Ying, Xi-xiang
author_facet Wang, Yun-jiao
Qu, Gong-lin
Zhang, Wen-jie
Xue, He-fei
Chen, Ying-hui
Yin, Jing-jing
Lu, Dong-rui
Ying, Xi-xiang
author_sort Wang, Yun-jiao
title Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
title_short Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
title_full Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
title_fullStr Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
title_full_unstemmed Pharmacokinetics, tissue distribution and excretion of Vitexin in mice
title_sort pharmacokinetics, tissue distribution and excretion of vitexin in mice
publishDate 2012
url http://sedici.unlp.edu.ar/handle/10915/25695
http://www.latamjpharm.org/resumenes/31/6/LAJOP_31_6_1_8.pdf
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