Pseudopolymorphism of Active Pharmaceutical Ingredients (APIs): A Case Study of L-Phenylalanine

The solid-state characterization, dimorphic nature, solubility and solvent-mediated transformation of the anhydrous form and the monohydrate form of L-phenylalanine have been firstly conducted in detail. The results have shown that, the two forms are enantiotropically related, and the transformatio...

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Autores principales: Lu, Jie, Liu, Zhen, Wang, Jing
Formato: Articulo
Lenguaje:Inglés
Publicado: 2012
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Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/18127
http://www.latamjpharm.org/resumenes/31/2/LAJOP_31_2_1_18.pdf
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Sumario:The solid-state characterization, dimorphic nature, solubility and solvent-mediated transformation of the anhydrous form and the monohydrate form of L-phenylalanine have been firstly conducted in detail. The results have shown that, the two forms are enantiotropically related, and the transformation rate can be prohibited by increasing temperature and reducing water content in the solvent mixtures. These results will contribute to a better understanding about the pseudopolymorphic systems for pharmaceutical industry.