Lipase-catalysed preparation of acyl derivatives of the germacranolide cnicin

Several acyl derivatives of cnicin were obtained through lipase-catalysed acylation and alcoholysis reactions. In most reactions lipases showed a regioselective behaviour affording only one product. Longer chain acyl derivatives were prepared at lower temperature than the used in lipase-catalysed re...

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Autor principal: Monsalve, L.N
Otros Autores: Rosselli, S., Bruno, M., Baldessari, A.
Formato: Capítulo de libro
Lenguaje:Inglés
Publicado: 2009
Acceso en línea:Registro en Scopus
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Registro en la Biblioteca Digital
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024 7 |2 scopus  |a 2-s2.0-68949122671 
024 7 |2 cas  |a cnicin, 24394-09-0; triacylglycerol lipase, 9001-62-1 
040 |a Scopus  |b spa  |c AR-BaUEN  |d AR-BaUEN 
030 |a JMCEF 
100 1 |a Monsalve, L.N. 
245 1 0 |a Lipase-catalysed preparation of acyl derivatives of the germacranolide cnicin 
260 |c 2009 
270 1 0 |m Baldessari, A.; Laboratorio de Biocatálisis, Departamento de Química Orgánica y UMYMFOR, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Pabellón 2, C1428EGA Buenos Aires, Argentina; email: alib@qo.fcen.uba.ar 
506 |2 openaire  |e Política editorial 
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520 3 |a Several acyl derivatives of cnicin were obtained through lipase-catalysed acylation and alcoholysis reactions. In most reactions lipases showed a regioselective behaviour affording only one product. Longer chain acyl derivatives were prepared at lower temperature than the used in lipase-catalysed reactions, to preclude side products formation. The enzymatic approach let to prepare a family of novel acetyl and fatty acid derivatives of cnicin which are not obtainable following traditional organic synthetic procedures. © 2008 Elsevier B.V. All rights reserved.  |l eng 
536 |a Detalles de la financiación: Agencia Nacional de Promoción Científica y Tecnológica, PICT 2005, 32735 
536 |a Detalles de la financiación: We thank UBA (project X089), ANPCyT (project PICT 2005, 32735) (Argentina) and Italian Government project PRIN for partial financial support. AB is a Research Member of CONICET. 
593 |a Laboratorio de Biocatálisis, Departamento de Química Orgánica y UMYMFOR, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Pabellón 2, C1428EGA Buenos Aires, Argentina 
593 |a Dipartimento di Chimica Organica, Università di Palermo, Viale delle Scienze, 90128 Palermo, Italy 
690 1 0 |a ACYLATION 
690 1 0 |a ALCOHOLYSIS 
690 1 0 |a CNICIN 
690 1 0 |a ENZYME CATALYSIS 
690 1 0 |a SESQUITERPENOIDS 
690 1 0 |a ACYL DERIVATIVES 
690 1 0 |a ALCOHOLYSIS 
690 1 0 |a ALCOHOLYSIS REACTIONS 
690 1 0 |a CNICIN 
690 1 0 |a ENZYME CATALYSIS 
690 1 0 |a FATTY ACID DERIVATIVES 
690 1 0 |a GERMACRANOLIDE 
690 1 0 |a REGIO-SELECTIVE 
690 1 0 |a SESQUITERPENOIDS 
690 1 0 |a SIDE PRODUCTS 
690 1 0 |a SYNTHETIC PROCEDURES 
690 1 0 |a ACYLATION 
690 1 0 |a ENZYMES 
690 1 0 |a FATTY ACIDS 
690 1 0 |a LIPASES 
690 1 0 |a CATALYSIS 
690 1 0 |a ACETIC ACID DERIVATIVE 
690 1 0 |a CNICIN 
690 1 0 |a FATTY ACID DERIVATIVE 
690 1 0 |a GERMACRANOLIDE DERIVATIVE 
690 1 0 |a SESQUITERPENE LACTONE 
690 1 0 |a TRIACYLGLYCEROL LIPASE 
690 1 0 |a UNCLASSIFIED DRUG 
690 1 0 |a ACYLATION 
690 1 0 |a ALCOHOLYSIS 
690 1 0 |a ARTICLE 
690 1 0 |a CATALYSIS 
690 1 0 |a CHEMICAL REACTION KINETICS 
690 1 0 |a CHEMICAL STRUCTURE 
690 1 0 |a CONTROLLED STUDY 
690 1 0 |a ENANTIOSELECTIVITY 
690 1 0 |a ENZYME ACTIVITY 
690 1 0 |a LOW TEMPERATURE 
690 1 0 |a NONHUMAN 
690 1 0 |a SYNTHESIS 
700 1 |a Rosselli, S. 
700 1 |a Bruno, M. 
700 1 |a Baldessari, A. 
773 0 |d 2009  |g v. 57  |h pp. 40-47  |k n. 1-4  |p J. Mol. Catal. B Enzym.  |x 13811177  |w (AR-BaUEN)CENRE-5687  |t Journal of Molecular Catalysis B: Enzymatic 
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856 4 0 |u https://doi.org/10.1016/j.molcatb.2008.06.019  |y DOI 
856 4 0 |u https://hdl.handle.net/20.500.12110/paper_13811177_v57_n1-4_p40_Monsalve  |y Handle 
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