Spectrofluorimetric assay for the photodegradation products of alprazolam

A new spectrofluorimetric assay for the photodegradation products of the ansiolytic drug alprazolam is described. Alprazolam was found to be highly photolabile and special care should be taken to avoid light exposure during alprazolam storage and handling. The photostability of alprazolam was evalua...

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Autor principal: Nudelman, N.S
Otros Autores: Gallardo Cabrera, C.
Formato: Capítulo de libro
Lenguaje:Inglés
Publicado: 2002
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PH
Acceso en línea:Registro en Scopus
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024 7 |2 cas  |a Alprazolam, 28981-97-7 
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030 |a JPBAD 
100 1 |a Nudelman, N.S. 
245 1 0 |a Spectrofluorimetric assay for the photodegradation products of alprazolam 
260 |c 2002 
270 1 0 |m Nudelman, N.S.; Depto. Quimica Organica, Facultad de Cie. Exactas y Natur., Universidad de Buenos Aires, 1428 Buenos Aires, Argentina; email: nudelman@qo.fcen.uba.ar 
506 |2 openaire  |e Política editorial 
504 |a Andrisano, V., Gotti, R., Leoni, A., Cavrini, V., (1999) J. Pharm. Biomed. Anal., 21, pp. 851-857 
504 |a Albini, A., Fasani, E., (1998) Drugs: Photochemistry and Photostability, pp. 1-73. , A. Albini, & E. Fasani. Cambridge: Royal Society of Chemistry 
504 |a Moore, D.E., (1996) Photostability of Drugs and Drug Formulations, pp. 9-38. , H.H. Tonnesen. London: Taylor and Francis 
504 |a Tonnesen, H.H., (1996) Photostability of Drugs and Drug Formulations, pp. 1-7. , H.H. Tonnesen. London: Taylor and Francis 
504 |a Piechocki, J.T., (1998) Drugs: Photochemistry and Photostability, pp. 247-271. , A. Albini, & E. Fasani. Cambridge: Royal Society of Chemistry 
504 |a Beijersbergen van Henegouwen, G.M.J., (1997) Adv. Drug Res., 29, pp. 79-170 
504 |a Wright, C.E., Sissin, T.L., Fleishaker, J.C., Antal, E.J., (1997) J. Clin. Pharmacol., 37, p. 321 
504 |a Nudelman, N.S., Waisbaum, R.G., (1997) J. Phys. Org. Chem., 10, pp. 97-106 
504 |a Nudelman, N.S., Waisbaum, R.G., (1995) J. Pharm. Sci., 84, pp. 208-211 
504 |a Nudelman, N.S., Waisbaum, R.G., (1995) J. Pharm. Sci., 84, pp. 998-1004 
504 |a Nudelman, N.S., Gallardo, C., (1999) Vitae, 6, pp. 29-40 
504 |a Nudelman, N.S., Waisbaum, R.G., Gallardo, C., (1998) Atualidades de Fisico-Quimica Organica, pp. 478-497 
504 |a Allen, L.E., Erickson, M.A., (1998) Am. J. Health Syst. Pharm., 55, pp. 1915-1920 
504 |a Caira, M.R., Easter, B., Honiball, S., Horne, A., Nassimbeni, L.R., (1995) J. Pharm. Sci., 84, pp. 1379-1384 
504 |a Andersin, R., Mesilaakso, M., (1995) J. Pharm. Biomed. Anal., 13, pp. 667-670 
504 |a Stemm, N.L., Skog, J.W., Robins, R.H., (1995) Pharm. Res., 12, pp. 738-745 
504 |a Cho, M.J., Scahill, T.A., Hester, J.B., (1983) J. Pharm. Sci., 72, pp. 356-362 
504 |a Konishi, M., Hirai, K., Mori, Y., (1982) J. Pharm. Sci., 71, pp. 1328-1334 
504 |a Jiménez, R.M., Dominguez, E., Baía, D., Alonso, R.M., Vicente, F., (1987) J. Heteroc. Chem., 24, pp. 421-424 
504 |a (1996) USP DI, 160 Edición, pp. 38-39 
504 |a Crouch, D.J., Rollins, D.E., Canfield, D.E., Andrenyak, D.M., Schulties, J.E., (1999) J. Anal. Toxicol., 23, pp. 479-485 
504 |a Hold, K.M., Rollins, D.E., Crouch, D.J., Wilkins, D.G., Canfield, D.E., Maes, R.A., (1996) J. Mass Spectrometry, 31, pp. 1033-1038 
504 |a Hall, M.A., Robinson, A., Brissie, R.M., (1995) J. Anal. Toxicol., 19, pp. 511-513 
504 |a Hold, K.M., Crouch, D.J., Rollins, D.E., Wilkins, D.G., Maes, R.A., (1997) Forensic Sci. Int., 84, pp. 201-209 
504 |a Hong, D.D., Shah, M., Drug Stability, Principles and Practices, 3 Edn., pp. 329-384. , J.T. Carstensen, C.T. Rhodes (ed.), Marcel Dekker Inc., New York 
504 |a Moore, D.E., (1996) Photostability of Drugs and Drug Formulations, pp. 63-82. , H.H. Tonnesen. London: Taylor and Francis 
504 |a Harth, Y., Rapoport, M., (1996) Drugs Sal., 14, pp. 252-259 
504 |a Reid, C.G., (1995) Can. Pharm. J., 128, pp. 31-56 
504 |a Harth, Y., Rapoport, M., (1996) Drugs Sal., 14, pp. 252-259 
504 |a Reid, C.G., (1995) Can. Pharm. J., 128, pp. 31-56 
504 |a Pazzagli, L., Banfi, R., Borselli, G., Semmola, M.V., (1998) Pharm. World Sci., 20, p. 136 
504 |a Watanabe, Y., Kawada, A., Ohnishi, Y., Tajima, S., Ishibashi, A., (1991) J. Am. Acad. Dermatol., 40, p. 832 
504 |a Kanwar, A.J., Gupta, R., Das Metha, S., (1990) Dermatologica, 181, p. 75 
504 |a Nudelman, N.S., Gallardo, C., (2002) J. Pharm. Sci., 91. , in press 
504 |a Minoru, O., Tsutomu, T., Toshihide, N., (1995) J. Pharm. Sci., 84, pp. 786-790 
520 3 |a A new spectrofluorimetric assay for the photodegradation products of the ansiolytic drug alprazolam is described. Alprazolam was found to be highly photolabile and special care should be taken to avoid light exposure during alprazolam storage and handling. The photostability of alprazolam was evaluated at pH 2.0, 3.6 and 5.0. The drug was exposed to UVA-UVB radiations, the photodegradation of alprazolam was followed by high-performance liquid chromatographic (HPLC) and the developed spectrofluorimetric assay allowed determination of the photodegradation products at very low concentrations (≥10-5 M). The photoinstability was found to increase with the pH value decreasing, consequently acidic media should be avoided during the drug-development process. © 2002 Elsevier Science B.V. All rights reserved.  |l eng 
536 |a Detalles de la financiación: Universidad de Buenos Aires 
536 |a Detalles de la financiación: Cancer Genomics Centre 
536 |a Detalles de la financiación: National Research Council 
536 |a Detalles de la financiación: Departamento Administrativo de Ciencia, Tecnología e Innovación, COLCIENCIAS 
536 |a Detalles de la financiación: Agency for Science, Technology and Research 
536 |a Detalles de la financiación: Consejo Nacional de Investigaciones Científicas y Técnicas 
536 |a Detalles de la financiación: CGC is a grateful recipient of a COLCIENCIAS fellowship. Financial support by the Agency for the Promotion of Science and Technology; the University of Buenos Aires and the National Research Council (CONICET) from Argentine is gratefully acknowledged. 
593 |a Depto. Quimica Organica, Facultad de Ciencias Exactas y Naturales, 1428 Buenos Aires, Argentina 
690 1 0 |a ALPRAZOLAM PHOTOSTABILITY 
690 1 0 |a ALPRAZOLAM QUALITY CONTROL 
690 1 0 |a ALPRAZOLAM STABILITY 
690 1 0 |a BENZODIAZEPINE PHOTOTOXICITY 
690 1 0 |a SPECTROFLUORIMETRIC ASSAY 
690 1 0 |a ALPRAZOLAM 
690 1 0 |a ARTICLE 
690 1 0 |a DRUG DEGRADATION 
690 1 0 |a DRUG DETERMINATION 
690 1 0 |a DRUG SCREENING 
690 1 0 |a DRUG STABILITY 
690 1 0 |a DRUG STORAGE 
690 1 0 |a FLUORESCENCE 
690 1 0 |a HIGH PERFORMANCE LIQUID CHROMATOGRAPHY 
690 1 0 |a LIGHT EXPOSURE 
690 1 0 |a PHOTODEGRADATION 
690 1 0 |a PRIORITY JOURNAL 
690 1 0 |a SPECTROFLUOROMETRY 
690 1 0 |a TABLET 
690 1 0 |a ULTRAVIOLET A RADIATION 
690 1 0 |a ULTRAVIOLET B RADIATION 
690 1 0 |a VALIDATION PROCESS 
690 1 0 |a ALPRAZOLAM 
690 1 0 |a DRUG STABILITY 
690 1 0 |a LIGHT 
690 1 0 |a SPECTROMETRY, FLUORESCENCE 
650 1 7 |2 spines  |a PH 
700 1 |a Gallardo Cabrera, C. 
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