Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes

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Biological and chemical characteristics of 99mTc‐phenethylamines complexes are presented. 2‐(4,5‐Dimethoxy‐2‐nitrophenyl)ethylamine, 2‐(3,4‐dimethoxyphenyl)ethylamine and 2‐(2‐amino‐4,5‐dimethoxyphenyl)‐ethylamine were used as ligands. A preliminary evaluation of these 99mTc‐complexes as dopamine re...

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Detalles Bibliográficos
Autor principal: Vitale, A.A
Otros Autores: Calvino, M.A, Ferrari, C.C, Stahl, A.E, Pomilio, A.B
Formato: Capítulo de libro
Lenguaje:Inglés
Publicado: 1995
Acceso en línea:Registro en Scopus
DOI
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Registro en la Biblioteca Digital
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Biblioteca Central Dr. Luis F. Leloir (FCEN) de Universidad de Buenos Aires
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100 1 |a Vitale, A.A. 
245 1 0 |a Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes 
260 |c 1995 
270 1 0 |m Vitale, A.A.; CONICET, Departamento de Química Orgánica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Ciudad Universitaria, Pabellón 2, Buenos Aires, 1428, Argentina 
506 |2 openaire  |e Política editorial 
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520 3 |a Biological and chemical characteristics of 99mTc‐phenethylamines complexes are presented. 2‐(4,5‐Dimethoxy‐2‐nitrophenyl)ethylamine, 2‐(3,4‐dimethoxyphenyl)ethylamine and 2‐(2‐amino‐4,5‐dimethoxyphenyl)‐ethylamine were used as ligands. A preliminary evaluation of these 99mTc‐complexes as dopamine receptor radioligands was also performed. Net charges at each atom were also calculated by a semiempirical ZINDO/1 method for comparison of free ligands' parameters with those of the respective technetium‐complexes. Copyright © 1995 John Wiley & Sons, Ltd.  |l eng 
593 |a CONICET, Departamento de Química Orgánica, Facultad de Ciencias Exactas y Naturales, Universidad de Buenos Aires, Ciudad Universitaria, Pabellón 2, Buenos Aires, 1428, Argentina 
593 |a Ineuci-Conicet, Departamento de Ciencias Biológicas, Fcen, Uba, Argentina 
690 1 0 |a 2‐(2‐AMINO‐4,5‐DIMETHOXYPHENYL)ETHYLAMINE 
690 1 0 |a 2‐(3,4‐DIMETHOXYPHENYL)‐ETHYLAMINE 
690 1 0 |a 2‐(4,5‐DIMETHOXY‐2‐NITROPHENYL)ETHYLAMINE 
690 1 0 |a 99M‐TECHNETIUM COMPLEXES 
690 1 0 |a BIODISTRIBUTION 
690 1 0 |a PREPARATION 
690 1 0 |a SEMIEMPIRICAL ZINDO/1 CALCULATIONS 
690 1 0 |a PHENETHYLAMINE DERIVATIVE 
690 1 0 |a TECHNETIUM 99M 
690 1 0 |a TECHNETIUM COMPLEX 
690 1 0 |a ANIMAL EXPERIMENT 
690 1 0 |a ARTICLE 
690 1 0 |a BRAIN 
690 1 0 |a CONTROLLED STUDY 
690 1 0 |a DRUG DISTRIBUTION 
690 1 0 |a DRUG STRUCTURE 
690 1 0 |a DRUG SYNTHESIS 
690 1 0 |a ELECTROPHORESIS 
690 1 0 |a FEMALE 
690 1 0 |a INTRACEREBRAL DRUG ADMINISTRATION 
690 1 0 |a ISOTOPE LABELING 
690 1 0 |a NONHUMAN 
690 1 0 |a RADIOCHROMATOGRAPHY 
690 1 0 |a RAT 
690 1 0 |a ANIMALIA 
700 1 |a Calvino, M.A. 
700 1 |a Ferrari, C.C. 
700 1 |a Stahl, A.E. 
700 1 |a Pomilio, A.B. 
773 0 |d 1995  |g v. 36  |h pp. 509-519  |k n. 6  |p J. Label. Compd. Radiopharm.  |x 03624803  |w (AR-BaUEN)CENRE-1949  |t Journal of Labelled Compounds and Radiopharmaceuticals 
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856 4 0 |u https://doi.org/10.1002/jlcr.2580360602  |y DOI 
856 4 0 |u https://hdl.handle.net/20.500.12110/paper_03624803_v36_n6_p509_Vitale  |y Handle 
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