Crystal packing modifies ligand binding affinity : The case of aldose reductase

The relationship between the structures of protein-ligand complexes existing in the crystal and in solution, essential in the case of fragment-based screening by X-ray crystallography (FBS-X), has been often an object of controversy. To address this question, simultaneous co-crystallization and soak...

Descripción completa

Guardado en:
Detalles Bibliográficos
Autores principales: Cousido-Siah, Alexandra, Petrova, Tatiana, Hazemann, Isabelle, Mitschler, André, Ruiz, Francesc X., Howard, Eduardo Ignacio, Ginell, Stepahn, Atmanene, Cédric, Van Dorsselaer, Alain, Sanglier-Cienférani, Sarah, Joachimiak, Andrzej, Podjarny, Alberto
Formato: Articulo Preprint
Lenguaje:Inglés
Publicado: 2012
Materias:
Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/96851
https://ri.conicet.gov.ar/11336/83350
https://onlinelibrary.wiley.com/doi/full/10.1002/prot.24136
http://europepmc.org/backend/ptpmcrender.fcgi?accid=PMC4671318&blobtype=pdf
https://www.ncbi.nlm.nih.gov/pubmed/22752989
Aporte de:

Ejemplares similares