QSPR modeling of the octanol/water partition coefficient of alcohols by means of optimization of correlation weights of local graph invariants

A particular approach based on the concept of flexible topological descriptors, the so called “Optimization of Correlation Weights of Local Graph Invariants”, is applied to model the octanol/water partition coefficient of a representative set of 62 alcohols. Predictions are quite satisfactory and th...

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Autores principales: Duchowicz, Pablo Román, Castro, Eduardo Alberto, Toropov, Andrey A.
Formato: Articulo
Lenguaje:Inglés
Publicado: 2004
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Acceso en línea:http://sedici.unlp.edu.ar/handle/10915/164019
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Sumario:A particular approach based on the concept of flexible topological descriptors, the so called “Optimization of Correlation Weights of Local Graph Invariants”, is applied to model the octanol/water partition coefficient of a representative set of 62 alcohols. Predictions are quite satisfactory and the numerical data improve previous results based on the application of a novel atomic-level-based AI topological descriptor. Some possible further extensions of the method are pointed out.